1996 – 2000

260.”A Facile Cleavage of Allyl Ethers on Solid Phase”
T. Opatz, H. Kunz, Tetrahedron Lett. 41 (2000), 10185-10188.

259.”The (2-Phenyl-2-trimethylsilyl)-ethoxycarbonyl(Psoc) Group ‚Äď a Novel Amino Protecting Group”
M. Wagner, S. Heiner, H. Kunz, Synlett  2000, 1753-1756

258.”Zur Entwicklung von Antitumor-Vakzinen: Ein synthetisches Konjugat aus tumorassoziiertem MUC1-Glycopeptidantigen und dem Tetanustoxin-Epitop”
S. Keil, C. Claus, W. Dippold, H. Kunz, Angew. Chem. 113 (2001), 379-382; Angew. Chem. Int. Ed. 40 (2001), 366-369

257.”Cyclodextrin-assisted Glycan Chain Extension on a Protected Glycosyl Amino Acid”
G. Dudziak, N. Bézay, T. Schwientek, H. Clausen, H. Kunz, A. Liese, Tetrahedron  56 (2000), 5865-5869

256.”Glycopeptide Synthesis in Solution and on Solid Phase”
H. Kunz, M. Schultz, in: Oligosaccharides in Chemistry and Biologogie РA Comprehensive Handbook ( B. Ernst, P. Sinay, G. W. Hart, Eds.), Wiley-VCH Verlag, Weinheim 2000, Bd. S  267-304

255.”Synthesis of Glycopeptides Containing Carbohydrate and Peptide Recognition Motifs”‚Ä®H. Herzner, T. Reipen, M. Schultz, H. Kunz,¬†Chem. Rev.¬†100 (2000), 4495-4537

254.”Streoselective Synthesis of 2-Substituted Pyrrolidines”
S. Deloisy, H. Tietgen, H. Kunz, Coll. Czechoslov. Chem. Commun. 65 (2000), 816-826

253.”Mixed Dialkylaluminum Chlorides and Mixed Trimethyl Organoaluminates in Chemoselective 1,4 Addition Reactions to Alkylidene Malonic Acid Diethyl ester”
S. Maas, H. Kunz, J. Prakt. Chem. 342 (2000), 396-403

252. “Glycosylation-induced asymmetric synthesis: b-amino acid esters via Mannich reaction”
P. Allef, H. Kunz, Tetrahedron Asymmetry 11 (2000), 375-378

251.”Synthesis of Sialyl Lewis A Glycopeptides ‚Äď A Partial Sequence of the P-Selectin Ligand PSGL-1″
K. Peilstöcker, H. Kunz, Synlett 2000, 823-825

250.”A Sialyl Lewis A-Building Block for Glycopeptide Synthesis”
K. Peilstöcker, H. Kunz, Synlett 2000, 820-822

249.”Synthetic Glycopeptide with Tumor-Associated Antigen and Cell Adhesion Ligand Structure”
H. Kunz, B. Liebe, O. Seitz, J. Habermann, K. Peilstöcker, U. Sprengard, in: Future Aspects in Peptide Chemistry  (W. Voelter, G. Fischer, Hrsg.) Collection Symposium Series  Vol. 1, 1999, 134-146

248.”Synthetic Glycopeptides and Glycoproteins”‚Ä®H. Kunz, in: Future Aspects in Peptide Chemistry¬† (W. Voelter, G. Fischer, Hrsg.) Collection Symposium Series¬† Vol. 1,¬†1999, 67-78

247.”Glycosylamines as Auxiliaries in Stereoselective Syntheses of Chiral Amino Compounds”
H. Tietgen, M. Schultz-Kukula, H. Kunz, in: Modern Amination Methods (A. Ricci, Hrsg.) Wiley-VCH Weinheim, 2000, 123-148

246.”Stereoselektive kombinatorische Ugi-Mehrkomponenten-Synthesen an fester Phase”‚Ä®K. Oertel, G. Zech, H. Kunz,¬†Angew. Chem. 112 (2000), 1489-1491,¬†Angew. Chem. Int. Ed. 39 (2000), 1431-1433

245. “Substituierte Tetrahydropyranderivate, Verfahren zu deren Herstellung, deren Verwendung als Arzneimittel oder Diagnostikum sowie sie enthaltendes Arzneimittel”
W. Schmitt, S. Henke, H. Kunz, C. Kallus, T. Opatz, T. Wunberg, Deutsche Patentanmeldung Hoechst Marion Roussel P197 34 392.9 vom 08.08.1997

244.”Chiral Auxiliaries in Cycloadditions”
K. R√ľck-Braun, H. Kunz, Wiley-VCH, Weinheim,¬†1999

243.”(2-Phenyl-2-trimethylsilyl)ethyl (PTMSE) Esters – A Novel Carboxyl Protecting Group”‚Ä®M. Wagner, H. Kunz,¬†Synlett¬†¬†2000, 400-402

242.”Combinatorial Solid-Phase Synthesis Using D-Galactose as a Chiral Five-Demensional-Diversity Scaffold”
Ch. Kallus, T. Opatz, T. Wunberg, W. Schmidt, S. Henke, H. Kunz, Tetrahedron Lett. 40 (1999), 7783-7786

241.”Selectively Deprotectable Carbohydrates Based on Regioselective Enzymatic Reactions”
R. Pfau, H. Kunz, Synlett 1999, 1817-1820

240.”Conjugate Addition of Dialkylaluminum Chlorides to Alkylidene Malonic Acid Derivatives”
S. Maas, A. Stamm, H. Kunz, Synthesis  1999, 1792-1798

239.”Mild Synthesis of Protected a-Glycosyl Iodides”
R. Caputo, H. Kunz, D. Mastroianni, G. Palumbo, S. Pedatella, F. Solla, Eur. J. Org. Chem. 1999, 3147-3150

238.”A Strategy towards the Stereoselective Synthesis of 5-Hydroxylysine”
B. Löhr, S. Orlich, H. Kunz, Synlett 1999, 139-141

237.”Modified Trityl Ester Protecting Groups in Peptide Synthesis”
B. Löhr, S. Orlich, H. Kunz, Synlett 1999, 136-138

236.”A Stereoselective Synthesis of Hydroxylysine and SPPS of a Glycosylated Collagen II Partial Structure”
B. Löhr, S. Orlich, H. Kunz, Peptides 1998 (Hrsg. S. Bajusz, F. Hudecz) Akademiai Kiado, Budapest 1999, 228-229

235.”Auxiliary-Controlled Stereoselective Enolate Protonation: Enantioselective Synthesis of cis and trans Annulated Decahydroquinoline Alkaloids”
M. Weymann, M. Schultz-Kukula, H. Kunz, Tetrahedron Lett. 39 (1998), 7835-7838

234.”Synthesis of Active Principles from the Leaves of Moringa oleifera Using S-Pent-4-enyl Thioglycosides”
M. Leuck, H. Kunz, Carbohydr. Res. 312 (1998), 33-44

233.”Desymmetrization Reactions on 4-Pyridone Using Carbohydrate Templates”
M. Follmann, H. Kunz, Synlett  1998 , 989-990

232. “Synthesis of Glycopeptides with Lewis antigen and Sialyl Lewis Antigen Side Chains”‚Ä®H. Kunz, K. von dem Bruch, G. Kretzschmar, U. Sprengard, in: Peptides, Biology and Chemistry, Proceedings of the 1996 Chinese Peptide Symposium (X.-J. Xu, Y.-H. Ye, J. P. Tam, Hrsg.), Kluwer Acad. Publ. Dordrecht 1998, 8-11

231.”Synthesis of Cyclic Dipeptide Templates, their Incorporation into Peptides and Studies on their Conformational and Biological Properties”
G. Asche, H. Kunz, H. Nar, H. Köppen, H. Briem, K.-H. Pook, P. W. Schiller, N. N. Chung, C. Lemieux, F. Escher, J. Peptide Res. 51 (1998) 323-336

230.”Kohlenhydrate als multfunktionelle chirale Ger√ľste in der kombinatorischen Synthese”‚Ä®T. Wunberg, C. Kallus, T. Opatz, S. Henke, W. Schmidt, H. Kunz,¬†Angew. Chem.¬†110 (1998), 2620-2622;Angew. Chem. Int. Ed. Engl. 37 (1998), 2503-2505.

229.”Stereoselective Syntheses of Chiral Heterocycles and Alkaloids Using Carbohydrate Auxiliaries”
H. Kunz, M. Weymann, M. Follmann, P. Allef, K. Oertel, M. Schultz-Kukula, A. Hofmeister, Polish J. Chem. 73 (1999), 15-27

228.”Effects of Glycosylation on Fragments of Tumor Associated Human Epithelial Mucin MUC1″
P. Braun, G. M. Davies, M. R. Price, P. M. Williams, S.J. B. Tendler, H. Kunz, Bioorg. Med. Chem. 6 (1998), 1531-1545

227.”Stereoselective Synthesis of Chiral Heterocycles Using Carbohydrates”
H. Kunz, M. Weymann, M. Follmann, C. Kallus, Chemické  listy  92 (1998) 258-260

226.”Carbhydrate Substituted Metallocenes as Chiral Complexes in Enantioselective Catalysis”
H. Kunz, A. Hofmeister, M. Puhl, Chemické  listy  92 (1998) 258

225.”Stereoselective Mannich Reaction with Tetrapivaloyl Galactosyl Bromide as Chiral Auxiliary”
H. Kunz. P. Allef, Chemické  listy  92 (1998) 257-258

224.”Fragment Condensation on Solid Phase in the Synthesis of an Amphiphlic Glycopeptide from the Homophilic Recognition Domain of Epithelial Cadherin 1‚ÄĚ
J. Habermann, H. Kunz, Tetrahedron Lett. 39 (1998) 4797-4800

223.”Enzymatic Hydrolysis of Hydrophilic Esters by Lipases in the Synthesis of Peptides and Glycopeptides”
M. Gewehr, P. Braun, O. Seitz, H. Kunz in: Peptides 1996  (Hrsg. R. Ramage, R. Epton), The European Peptide Society 1998, Mayflower Scietific Ltd. Kingswinford, 421-422

222.”Allylic Anchoring Groups in Solid Phase Synthesis”
N. Bezay, G. Fuchs, J. Habermann, B. Liebe, B. Löhr, O. Seitz, H. Kunz in: Peptides 1996 (Hrsg. R. Ramage, R. Epton), The European Peptide Society 1998, Mayflower Scietific Ltd. Kingswinford, 257-258

221.”Glycopeptide Synthesis Using O-Pentafluorophenyluronium Salts as Novel Condensing Reagents”
J. Habermann, H. Kunz, J. prakt. Chem. 340 (1998) 233-239

220.”A Novel Synthesis of Chain-Extended Amino Sugar Derivatives through Aza-Cope Rearrangement of N-Galactosyl N-Homoallylamines”
S. Deloisy, H. Kunz, Tetrahedron Lett. 39 (1998) 791-794

219.”Solid-Phase Synthesis of a Glycopeptide from the Homophilic Recognition Domain of Epithelial Cadherin 1 Using a O-Pentafluorophenyluronium Salt”
J. Habermann, H. Kunz, Tetrahedron Lett. 39 (1998), 265-268

218.”Enantioselective Allylic Substitution Using a Novel (Phosphino-a-D-glucopyrano-oxazo-line)Palladium Catalyst”
B. Gläser, H. Kunz, Synlett  1998, 53-54

217.”Oligosaccharide Synthesis via Electrophile-induced Activation of Glycosyl-N-allylcarbamates”
H. Herzner, J. Eberling M. Schultz, J. Zimmer, H. Kunz, J. Carbohydr. Chem. 17 (1998) 759-776

216.”Pentafluorophenyluronium Reagents and Allylic Anchoring Groups in Solid Phase Glycopeptide Synthesis”
J. Habermann, H. Kunz, in: Solid Phase Synthesis and Combinatorial Chemical Libraries (1999) (Hrsg. R. Epton), Mayflower Worldwide Ltd., Birmingham, U. K., (1999), 217-220

215.”Recent Advances in the Synthesis of Glycopeptides”
H. Kunz, M. Schultz in: Glycopeptides and Related Compounds (Hrsg. D. G. Large, C. D. Warren), Marcel Dekker, New York 1997, 23-78

214.”Stereoselective Synthesis Using Carbohydrates as Carriers of Chiral Information”
H. Kunz, A. Hofmeister, B. Gläser in: Polysaccharides. Structural Diversity and Functional Versatility  (Hrsg. S. Dumitriu), Marcel Dekker, New York, 1998, 539-567

213.”Chemistry of Glycopeptides”
H. Kunz, B. Löhr, J. Habermann in Carbohydrates: Structure, Dynamics and Synthesis (Hrsg: P. Finch), Kluwer Academic Publishers, Dordrecht 1999, p 187-227

212.”Comparative Lipase-catalyzed Hydrolysis of Ethylene-glycol-derived Esters. – The 2-Methoxyethyl Ester as Protective Group in Peptide and Glycopeptide Synthesis”
M. Gewehr, H. Kunz, Synthesis 1997, 1499-1511

211.”Solid-Phase Synthesis of a Sialyl-Tn-Glycoundecapeptide of the MUC-1 Repeating Unit”
B. Liebe, H. Kunz, Helv. Chim. Acta  80 (1997) 1473-1482

210.”Enantioselective Synthesis of 2-Alkyl-, 2,6-Dialkylpiperidine, and Indolizidine-Alkaloids through Diastereoselective Mannich-Michael Reaction Cascades”
M. Weymann, W. Pfrengle, D. Schollmeyer, H. Kunz, Synthesis  1997, 1151-1160

209.”Use of the Allylic HYCRON Anchor in Solid Phase Peptide Synthesis”
M. Gewehr, H. Kunz, A. Lauterbach, B. L√∂hr, O. Seitz in “Innovation and Perspectives in Solid Phase Synthesis 1996″ (Hrsg. R. Epton), Mayflower Scientific Ltd., Birmingham,¬†1997, 117-120

208.”Neue Dipeptidtemplate, Verfahren zu deren Herstellung und deren Verwendung zum Einbau in Peptidsequenzen, unter anderem auf dem Gebiet der kombinatorischen Chemie”‚Ä®F. Esser, G. Asche, H. Kunz, Deutsche Patentanmeldung P 197 03 801.8 (Boehringer Ingelheim KG) 1. 2. 1997

207.”Synthesis of TN and T Antigen Glycopeptide Sequences of Tumor-Associated MUC-1 Using S-Pentenyl Thioglycosides”
M. Leuck, H. Kunz, J. prakt. Chem. 339 (1997), 332-334

206.”Festphasensynthese eines tumorassoziierten Sialyl-Tn-Antigen-Glycopeptids mit einer Partialsequenz aus dem “Tandem Repeat” des MUC-1-Mucins”
B. Liebe, H. Kunz, Angew. Chem. 109 (1997), 629-631; Angew. Chem. Int. Ed. Engl. 36 (1997), 618-621

205.”N,N,N’,N’-Tetrasubstituierte O-Pentafluorphenyl-Uroniumsalze als neue Kondensations-reagenzien zu Synthesen von Amiden und speziell Peptiden”
H. Kunz, J. Habermann, Deutsche Patentanmeldung  196 48 125.2 (21.11. 1996)

204.”HYCRON – An Allylic Anchor for High-Efficiency Solid-Phase Synthesis of Protected Peptides and Glycopeptides”
O. Seitz, H. Kunz, J. Org. Chem. 62 (1997), 813-826

203.”b-Branched a-Halocarboxylic Acid Derivatives via Stereoselective 1,4 Addition of Dialkylaluminum Chlorides to a,b-Unsaturated N-Acyl Oxazolidinones”
K. R√ľck-Braun, A. Stamm, S. Engel, H. Kunz, J. Org. Chem. 62 (1997), 967-975

202.”Synthesis and Biological Activity of Novel Sialyl-Lewisx Conjugates”
U. Sprengard, H. Kunz, C. H√ľls, W. Schmidt, D. Seiffge, G. Kretzschmar,¬†Bioorg. Med. Chem. Lett.¬†6 (1996), 509-514

201.”Glycosyl Azides as Building Blocks in Convergent Syntheses of Oligomeric Lactosamine and Lewisx Saccharides”
W. Bröder, H. Kunz, Bioorg. Med. Chem. 5 (1997), 1-19

200.”Asymmetrische Mannich-Synthese von b-Aminos√§uren mit zwei neuen stereogenen Zentren in a- und b-Position”
H. Kunz, A. Burgard, D. Schanzenbach, Angew. Chem. 109 (1997), 394-396; Angew. Chem. Int. Ed. Engl. 36 (1997), 386-387

199.”Chemoselective Removal of Protecting Groups from O-Glycosyl Amino Acid and Peptide Methoxyethoxyethyl Ethers Using Lipases and Papain”
J. Eberling, P. Braun, D. Kowalczyk, M. Schultz, H. Kunz, J. Org. Chem. 61 (1996), 2638-2646

198. “Solid-Phase Synthesis of a 36 Amino Acid O-Fucosyl-Peptide with the Uncommon Thr-Fuc Linkage”
H. Hietter, M. Schultz, H. Kunz, Synlett 1995, 1219-1220

197.”Synthetic Tumor-Associated Glycopeptide Antigens”
O. Seitz, B. Liebe, P. Braun, K. von dem Bruch, H. Kunz in “Control Mechanisms of Cancinogenesis” (Ed. J. Hengstler, F. Oesch), Institut f√ľr Toxikologie, Mainz,¬†1996, S. 338- 354

196.”Synthetic Glycopeptides and Neoglycoproteins of Biological Interest”
H. Kunz in “Peptides in Immunology” (Hrsg. C. H. Schneider) J. Wiley and Sons Ltd, Chichester¬†1996, 9-17

195.”Oligosaccharide Recognition by Selectins: Synthesis and Biological Activity of Multivalent Sialyl Lewis-X Ligands”
G. Kretzschmar, U. Sprengard, H. Kunz, E. Bartnik, W. Schmidt, A. Toepfer, B. Hörsch, M. Krause, D. Seiffge,Tetrahedron 51 (1995), 13015-13030

194.”Carbohydrates as Chiral Templates in the Stereoselective Synthesis of b-Amino Acids”‚Ä®H. Kunz, M. Weymann, A. Burgard, in “Enatioselective Synthesis of b-Amino Acids” (Eusebio Juaristi, Hrsg.), Wiley-VCH Publ., New York, 1997, S. 407-422

193.”Multiple Sialyl-Lewisx-N-Glycopeptide:Effektive Liganden f√ľr E-Selektin”
U. Sprengard, M. Schudok, G. Kretzschmar, H. Kunz, Angew. Chem. 108 (1996), 359-362. Angew. Chem. Int. Ed. Engl. 35 (1996), 321-324